SCHEMBL27925516

SCHEMBL27925516

O=C(O)c1cc(OC(F)CF)nn1-c1ncccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCK P35557 11/20 0.35
KCNH2 Q12809 5/20 0.34
TRPA1 O75762 3/20 0.33
HIF1A Q16665 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
MALT1 Q9UDY8 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27944900 0.91 GCK (0.33) GCKKCNH2TRPA1TRPV1MALT1
SCHEMBL14658369 0.89 GCK (0.34) GCKKCNH2TRPA1TRPV1MALT1
SCHEMBL16014740 0.89 NPC1 (0.37) GCKKCNH2TRPA1TRPV1MALT1
SCHEMBL16014767 0.84 TRPA1 (0.36) GCKKCNH2TRPA1HIF1ATRPV1
SCHEMBL16014575 0.84 ALDH1A1 (0.39) GCKKCNH2TRPA1MALT1
SCHEMBL27944843 0.83 P2RX7 (0.34)
SCHEMBL29185079 0.83 TRPA1 (0.35) GCKKCNH2TRPA1TRPV1MALT1
SCHEMBL27962696 0.81 ALDH1A1 (0.40) GCKTRPA1TRPV1MALT1KMT2A
SCHEMBL16014505 0.81 NPC1 (0.40) GCKKCNH2TRPA1HIF1A
SCHEMBL14658366 0.80 TRPA1 (0.36) TRPA1HIF1ATRPV1MALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103130769-B 3-difluoro ethoxy-pyrazole amides compounds and application thereof UNIV QINGDAO SCIENCE & TECHNOLOGY 2014-12-17 CN disclosed
CN-103420975-A Fluorine-contained o-amino thiobenzamide type compound and application thereof UNIV QINGDAO SCIENCE & TECHNOLOGY 2013-12-04 CN disclosed
CN-103130769-A 3-difluoro ethoxy-pyrazole amides compounds and application thereof UNIV QINGDAO SCIENCE & TECHNOLOGY 2013-06-05 CN disclosed