SCHEMBL27933705

SCHEMBL27933705

Cc1nnn(-c2ccc(F)cc2)c1-c1cn(-c2ccc(C(C)C(=O)C(C)c3ccc(-n4cnc(-c5c(C)nnn5-c5ccc(F)cc5)c4)cc3)cc2)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.39
GABRA5 P31644 5/20 0.36
MAPK1 P28482 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
SLC5A1 P13866 1/20 0.35
SLC5A2 P31639 1/20 0.35
LMNA P02545 3/20 0.35
NPC1 O15118 2/20 0.35
MAPT P10636 2/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9895210 0.84 PTGS2 (0.46) PTGS2GABRA5LMNANPC1TSHR
SCHEMBL28807048 0.81 PTGS2 (0.39) PTGS2GABRA5SLC5A1SLC5A2LMNA
SCHEMBL27933718 0.80 MAPK1 (0.35) GABRA5MAPK1PSEN1PSEN2APH1B
SCHEMBL9895924 0.79 RAB9A (0.38) PTGS2IDO1TDO2LMNANPC1
SCHEMBL9896578 0.76 LMNA (0.38) PTGS2LMNANPC1RAB9ABRD4
SCHEMBL21402163 0.76 PTGS2 (0.40) PTGS2GABRA5LMNAGAAL3MBTL1
SCHEMBL9895133 0.75 GABRA5 (0.43) GABRA5MAPTBRD4BRD2BRD3
SCHEMBL9895805 0.75 MAP4K4 (0.38) PTGS2NPC1TSHRRAB9ABRD4
SCHEMBL9894949 0.73 RAB9A (0.40) PTGS2GABRA5IDO1TDO2NPC1
SCHEMBL27915203 0.73 PTGS2 (0.52) PTGS2GABRA5IDO1TDO2SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249728-A Novel triazole compounds III HOFFMANN LA ROCHE 2013-08-14 CN claimed
CN-103249728-A Novel triazole compounds III HOFFMANN LA ROCHE 2013-08-14 CN disclosed