SCHEMBL27936769

SCHEMBL27936769

CC(=O)Oc1c(-c2cccc(OC(F)(F)F)c2)noc1C

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.45
PTGS2 P35354 1/20 0.43
GRM5 P41594 1/20 0.42
POLB P06746 1/20 0.40
POLQ O75417 1/20 0.39
KCNK3 O14649 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
S1PR1 P21453 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27918183 0.87 XDH (0.44) GPBAR1GRM5POLQKCNK3S1PR1
SCHEMBL28805571 0.85 GPBAR1 (0.46) GPBAR1PTGS2POLBNTRK1
SCHEMBL27936779 0.83 GPBAR1 (0.55) GPBAR1POLB
SCHEMBL27918191 0.82 GPBAR1 (0.53) GPBAR1
SCHEMBL13732600 0.81 GPBAR1 (0.51) GPBAR1PTGS2POLBCSNK2A2CSNK2B
SCHEMBL13735662 0.80 GPBAR1 (0.52) GPBAR1PTGS2POLB
SCHEMBL27495331 0.78 KMT2A (0.55) GPBAR1PTGS2POLB
SCHEMBL27936773 0.78 GABRA5 (0.45) GPBAR1PTGS2NTRK1
SCHEMBL2777083 0.78 TDP1 (0.53) GPBAR1PTGS2POLB
SCHEMBL28805573 0.76 ALDH1A1 (0.46) GPBAR1S1PR1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103313982-B Phenyl-isoxazole derivatives and process for the preparation thereof IL-YANG PHARM. CO.,LTD. (KR) 2016-02-03 CN disclosed
CN-103313982-A Phenyl-isoxazole derivatives and process for the preparation thereof IL YANG PHARM CO LTD 2013-09-18 CN disclosed