SCHEMBL27937992

SCHEMBL27937992

O=C(c1cc(=O)c2ccccc2o1)N1CCOCC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.65
LMNA P02545 2/20 0.63
HTT P42858 2/20 0.63
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
HSD17B10 Q99714 1/20 0.63
PRKDC P78527 2/20 0.58
ACE P12821 1/20 0.58
ECE1 P42892 1/20 0.58
KDM4E B2RXH2 3/20 0.57
USP2 O75604 1/20 0.57
CSNK2A2 P19784 1/20 0.57
PTGS1 P23219 1/20 0.57
CSNK2B P67870 1/20 0.57
CSNK2A1 P68400 1/20 0.57
CSNK2A3 Q8NEV1 1/20 0.57
ALDH1A1 P00352 7/20 0.57
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1942279 0.85 POLB (0.71) POLBLMNAHTTMEN1KMT2A
SCHEMBL7086091 0.85 POLB (0.63) POLBLMNAHTTMEN1KMT2A
SCHEMBL1946681 0.83 RAB9A (0.70) POLBLMNAHTTMEN1KMT2A
SCHEMBL1945801 0.83 ALDH1A1 (0.60) POLBLMNAHTTMEN1KMT2A
SCHEMBL18889298 0.81 MAPT (0.78) POLBLMNAMEN1KMT2ANPSR1
SCHEMBL5584787 0.81 RAB9A (0.53) POLBLMNAHTTMEN1KMT2A
SCHEMBL20886734 0.80 KMT2A (0.50) POLBHTTMEN1KMT2AKDM4E
SCHEMBL1941907 0.79 ALDH1A1 (0.74) POLBLMNAHTTMEN1KMT2A
SCHEMBL1944863 0.77 RAB9A (0.70) POLBLMNAHTTMEN1KMT2A
SCHEMBL1943197 0.75 ALDH1A1 (0.78) POLBLMNAHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103596948-B Benzopyranone compounds as PI 3-kinase inhibitors for the treatment of cancer ASTRAZENECA AB (SE) 2016-04-27 CN disclosed
CN-103596948-A Benzopyranone compounds as PI 3-kinase inhibitors for the treatment of cancer ASTRAZENECA AB 2014-02-19 CN disclosed