SCHEMBL27939656

SCHEMBL27939656

CCC(Oc1cc(N)ccc1OC)N(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.49
KDM4E B2RXH2 5/20 0.49
MAPT P10636 4/20 0.49
HTT P42858 2/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP19A1 P11511 2/20 0.41
NR4A1 P22736 1/20 0.41
ALDH1A1 P00352 5/20 0.39
USP2 O75604 2/20 0.39
LMNA P02545 1/20 0.38
ATM Q13315 2/20 0.37
AOC3 Q16853 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
CASP1 P29466 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404286 0.79 KDM4E (0.45) GAAKDM4EMAPTHTTTSHR
SCHEMBL8687840 0.75 KDM4E (0.45) GAAKDM4EMAPTHTTTSHR
SCHEMBL1010304 0.74 KDM4E (0.50) GAAKDM4EMAPTHTTTSHR
SCHEMBL8388931 0.73 KDM4E (0.50) GAAKDM4EMAPTHTTTSHR
SCHEMBL77823 0.73 KDM4E (0.67) GAAKDM4EMAPTHTTTSHR
SCHEMBL29377777 0.73 KDM4E (0.67) GAAKDM4EMAPTHTTTSHR
SCHEMBL2438047 0.73 KDM4E (0.67) GAAKDM4EMAPTHTTTSHR
SCHEMBL4323659 0.73 KDM4E (0.49) GAAKDM4EMAPTHTTTSHR
SCHEMBL18727243 0.72 KDM4E (0.57) GAAKDM4EMAPTHTTTSHR
SCHEMBL7502802 0.72 ALDH1A1 (0.57) GAAKDM4EMAPTHTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103626761-B Benazepine compound and the application as antitumor drug thereof SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2015-07-29 CN disclosed
CN-103626761-A Benazepine compound and application thereof as antitumor drug CISEN PHARMACEUTICAL CO LTD 2014-03-12 CN disclosed