SCHEMBL27951817

SCHEMBL27951817

CC(=O)c1csc(Cn2n[c]cn2)n1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
KDM1A O60341 5/20 0.35
HRH3 Q9Y5N1 2/20 0.34
FPR2 P25090 7/20 0.33
FPR3 P25089 6/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP13 P45452 1/20 0.33
PTGER1 P34995 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704174 0.74 MAPT (0.40) MAPTNPC1RAB9AKDM1AHRH3
SCHEMBL2332615 0.73 MAPT (0.40) MAPTNPC1RAB9AKDM1AHRH3
SCHEMBL27939524 0.72 RAB9A (0.37) NPC1RAB9AFPR2FPR3
SCHEMBL28810508 0.72 ALDH1A1 (0.36) MAPTNPC1RAB9AMMP13
SCHEMBL2818990 0.70 MAPT (0.42) MAPTNPC1RAB9AKDM1AHRH3
SCHEMBL1703731 0.70 MAPT (0.38) MAPTNPC1RAB9AHRH3FPR2
SCHEMBL13547516 0.70 MAPT (0.53) MAPTNPC1RAB9AKDM1AFPR2
SCHEMBL8280912 0.70 HRH3 (0.63) MAPTNPC1RAB9AHRH3FPR2
SCHEMBL2642294 0.69 MAPT (0.51) MAPTNPC1RAB9AKDM1AFPR2
SCHEMBL9926020 0.69 MAPT (0.51) MAPTNPC1RAB9AKDM1AFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101903378-B Aminotriazole derivatives ACTELION PHARMACEUTICALS LTD 2014-03-12 CN claimed
CN-101903378-B Aminotriazole derivatives ACTELION PHARMACEUTICALS LTD 2014-03-12 CN disclosed