SCHEMBL27955445

SCHEMBL27955445

Cc1ccccc1N1CCNCC1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.47
HTR2C P28335 11/20 0.47
HTR2B P41595 9/20 0.47
HTR2A P28223 5/20 0.47
ITGB1 P05556 2/20 0.42
ITGA5 P08648 2/20 0.42
MAPT P10636 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
ITGA4 P13612 1/20 0.41
TACR1 P25103 1/20 0.41
HTR7 P34969 1/20 0.40
TSHR P16473 1/20 0.40
AR P10275 1/20 0.39
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3645088 0.81 TACR1 (0.46) HTR2CHTR2BHTR2ATACR1HTR6
SCHEMBL5384916 0.81 TACR1 (0.59) HTR2CHTR2BHTR2ATACR1HTR7
SCHEMBL20140971 0.80 SLC6A2 (0.53) ADRB1HTR2CHTR2BHTR2ATSHR
SCHEMBL9396845 0.80 SLC6A2 (0.53) ADRB1HTR2CHTR2BHTR2ATSHR
Hydrochloric Acid SCHEMBL20140710 0.79 SLC6A2 (0.51) ADRB1HTR2CHTR2BHTR2ATSHR
SCHEMBL29977101 0.79 HTR1A (0.60) ADRB1HTR2CHTR2AHTR7HTR6
SCHEMBL28907620 0.79 HTR1A (0.60) ADRB1HTR2CHTR2AHTR7HTR6
SCHEMBL28081734 0.78 ITGB3 (0.53) ITGB1ITGA5MAPTITGB3ITGAV
SCHEMBL2877579 0.77 ADRB1 (0.54) ADRB1HTR2CHTR2BHTR2AHTR7
SCHEMBL21268736 0.77 ADRB1 (0.54) ADRB1HTR2CHTR2BHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101778831-B piperazine amide derivatives HOFFMANN LA ROCHE 2014-08-20 CN disclosed
CN-103772299-A Novel piperazine amide derivatives HOFFMANN LA ROCHE 2014-05-07 CN disclosed