SCHEMBL27974641

SCHEMBL27974641

CN(C)C(Cl)C(=O)c1cccc(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
CHRNB2 P17787 1/20 0.49
SLC6A2 P23975 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
SLC6A3 Q01959 1/20 0.49
PARP1 P09874 1/20 0.49
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
OPRM1 P35372 1/20 0.45
OPRL1 P41146 1/20 0.45
PLA2G7 Q13093 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4435825 0.81 CES2 (0.54) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL3269025 0.80 CES2 (0.61) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL29281060 0.79 CES2 (0.59) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL28036133 0.78 RAB9A (0.49) CES2CES1NPC1RAB9AMEN1
SCHEMBL8400060 0.77 PARP1 (0.58) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL28075891 0.77 CES2 (0.57) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL28748136 0.77 CES2 (0.57) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL3362925 0.77 CES2 (0.61) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL8015553 0.77 CES2 (0.61) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL28238806 0.76 CES2 (0.56) CES2CES1CHRNB2SLC6A2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965161-A Substituted 2-aminopyridine inhibitor for protein kinase CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD 2014-08-06 CN disclosed
CN-103965168-A Aryl/heteroaryl-substituted 2-aminopyridine inhibitor for protein kinase CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD 2014-08-06 CN disclosed