SCHEMBL2797668

SCHEMBL2797668

COC(=O)c1ccc([N+](=O)[O-])c(O)c1.O=C(O)c1ccc([N+](=O)[O-])c(O)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.58
CASP6 P55212 1/20 0.57
TSHR P16473 2/20 0.56
VCAM1 P19320 1/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA7 P43166 1/20 0.54
XDH P47989 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
HCAR3 P49019 5/20 0.52
MAPT P10636 3/20 0.49
LMNA P02545 2/20 0.49
MEN1 O00255 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29433264 0.94 XDH (0.61) TPMTVCAM1CA12CA1CA2
SCHEMBL223930 0.94 XDH (0.61) TPMTVCAM1CA12CA1CA2
SCHEMBL459609 0.87 CASP6 (0.72) TPMTCASP6TSHRCA12CA1
SCHEMBL31011353 0.87 CASP6 (0.72) TPMTCASP6TSHRCA12CA1
SCHEMBL2797670 0.85 MAPT (0.51) TPMTVCAM1CA12CA1CA2
SCHEMBL1353346 0.82 VCAM1 (0.57) CASP6TSHRVCAM1HCAR3LMNA
SCHEMBL2722165 0.82 CASP6 (0.60) CASP6TSHRVCAM1HCAR3MAPT
SCHEMBL31548461 0.82 CASP6 (0.60) CASP6TSHRVCAM1HCAR3MAPT
SCHEMBL531728 0.81 VCAM1 (0.64) TPMTTSHRVCAM1CA12CA1
SCHEMBL5734347 0.81 VCAM1 (0.68) CASP6VCAM1MAPTLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393782-A1 BENZOIC ACID (1-PHENYL-2-PYRIDIN-4-YL) ETHYL ESTERS AS PHOSPHODIESTERASE INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2011-12-14 EP disclosed
WO-2010089107-A1 BENZOIC ACID (1-PHENYL-2-PYRIDIN-4-YL) ETHYL ESTERS AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2010-08-12 WO disclosed