SCHEMBL28814538

SCHEMBL28814538

Nc1nc(N)c(-c2cnccn2)c(-c2nn[nH]n2)n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
CYP2A6 P11509 1/20 0.36
GLA P06280 1/20 0.33
PPARA Q07869 1/20 0.33
P2RX3 P56373 1/20 0.32
P2RX2 Q9UBL9 1/20 0.32
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27850416 0.76 HSP90AA1 (0.43) KDM4EGLA
SCHEMBL27985753 0.75 DHFR (0.33) KDM4EGLA
Hydrochloric Acid SCHEMBL1367779 0.75 HSP90AA1 (0.41) KDM4EGLA
SCHEMBL27985752 0.73 ADORA2A (0.44) KDM4EGLA
SCHEMBL27985443 0.72 KDM4E (0.46) KDM4ECYP2A6
SCHEMBL27831916 0.72 PIM1 (0.36) KDM4EGLA
SCHEMBL28791336 0.71 ADORA2A (0.48) CYP2A6
SCHEMBL27985373 0.71 DHFR (0.37) KDM4EGLAPPARA
SCHEMBL28814482 0.70 ADORA2A (0.47) KDM4ECYP2A6GLA
SCHEMBL27985802 0.70 PIK3CD (0.35) KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN claimed
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN disclosed