SCHEMBL28000258

SCHEMBL28000258

CN1CCN(c2cccc(NC(=O)O)c2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.64
HTR1D P28221 2/20 0.64
HTR1B P28222 2/20 0.64
KDM1A O60341 1/20 0.58
RCOR1 Q9UKL0 1/20 0.58
CASP3 P42574 1/20 0.57
CASP7 P55210 1/20 0.57
SETD2 Q9BYW2 1/20 0.57
MEN1 O00255 3/20 0.55
USP2 O75604 3/20 0.55
MAPT P10636 3/20 0.55
KMT2A Q03164 3/20 0.55
POLB P06746 2/20 0.55
MAPK1 P28482 2/20 0.55
HCRTR1 O43613 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
HTT P42858 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30577378 0.88 HTR1D (0.60) HTR2AHTR1DHTR1BKDM1ARCOR1
SCHEMBL22410915 0.87 HTR2A (0.59) HTR2AHTR1DHTR1BKDM1ARCOR1
SCHEMBL25319314 0.86 MAPT (0.68) HTR2AHTR1DHTR1BMEN1USP2
SCHEMBL22169759 0.84 BRD4 (0.58) HTR2AHTR1DHTR1BKDM1ARCOR1
SCHEMBL19281787 0.84 FAAH (0.52) HTR2AHTR1DHTR1BMEN1USP2
SCHEMBL16583818 0.82 KMO (0.61) CASP3CASP7SETD2MEN1USP2
SCHEMBL29521619 0.82 HTR2A (0.52) HTR2AHTR1DHTR1BKDM1ARCOR1
SCHEMBL20557362 0.81 CNR1 (0.79) HTR2AHTR1DHTR1BMEN1USP2
SCHEMBL30469240 0.81 CNR1 (0.79) HTR2AHTR1DHTR1BMEN1USP2
SCHEMBL28106923 0.81 RAB9A (0.70) MEN1MAPTKMT2APOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104684554-A Derivatives of azaindazole or diazaindazole type for treating pain PF MEDICAMENT 2015-06-03 CN disclosed
CN-104470925-A Imidazotriazinecarbonitriles useful as kinase inhibitors BRISTOL MYERS SQUIBB CO 2015-03-25 CN disclosed