SCHEMBL2800092

SCHEMBL2800092

CCC(C(=O)O)n1c(=O)cc(C)c2ccc(OC)cc21

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.42
AKR1C2 P52895 3/20 0.42
AKR1C1 Q04828 1/20 0.42
PTGS1 P23219 1/20 0.42
KDM4E B2RXH2 8/20 0.42
ALDH1A1 P00352 4/20 0.42
HSD17B10 Q99714 3/20 0.42
HPGD P15428 2/20 0.42
MAPK1 P28482 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 1/20 0.41
ATM Q13315 1/20 0.41
PLA2G10 O15496 1/20 0.40
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11191901 0.79 NPC1 (0.44) AKR1C3AKR1C2KDM4EALDH1A1HSD17B10
SCHEMBL5040312 0.76 KDM4E (0.64) KDM4E
SCHEMBL12002162 0.75 KDM4E (0.56) KDM4EALDH1A1HSD17B10HPGDMAPK1
SCHEMBL2953262 0.74 KMO (0.60) AKR1C3AKR1C2AKR1C1PTGS1KDM4E
SCHEMBL13234297 0.73 KDM4E (0.69) KDM4EALDH1A1HSD17B10MAPK1TSHR
SCHEMBL392780 0.73 NQO2 (0.57) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL2798839 0.73 POLB (0.52) ALDH1A1SMN1; SMN2
SCHEMBL2800556 0.72 AKR1C3 (0.43) AKR1C3AKR1C2
SCHEMBL2797974 0.72 CCNE2 (0.47) KDM4EALDH1A1HSD17B10HPGDMAPK1
SCHEMBL2955732 0.72 KMO (0.51) AKR1C3AKR1C2AKR1C1PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329694-B2 Quinoxalinones as antibacterial composition TOYAMA CHEMICAL CO., LTD. (JP) 2012-12-11 US disclosed
US-20100168418-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2010-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168418-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF ROS1, NOX1, ARG1 AKR1C3 976/4885AKR1C2 1542/4885AKR1C1 1133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.