Biphenyl

Biphenyl

SCHEMBL2800407

CS(=O)(=O)Nc1ccncc1.c1ccc(-c2ccccc2)cc1

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.64
CYP17A1 P05093 1/20 0.52
USP2 O75604 1/20 0.52
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP2C19 P33261 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
PGR P06401 1/20 0.51
PTGS2 P35354 3/20 0.51
PTGS1 P23219 2/20 0.51
KIF11 P52732 3/20 0.50
NR3C2 P08235 3/20 0.50
NOTUM Q6P988 1/20 0.50
MAPK10 P53779 1/20 0.49
KDM1A O60341 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423573 0.88 KEAP1 (0.60) KEAP1LMNAPGRPTGS2PTGS1
SCHEMBL873846 0.84 KEAP1 (0.75) KEAP1LMNAPGRPTGS2KIF11
SCHEMBL56693 0.80 KEAP1 (1.00) KEAP1LMNAPGRPTGS2KIF11
SCHEMBL18427042 0.78 KEAP1 (0.64) KEAP1LMNAPGRPTGS2KIF11
Hydrochloric Acid SCHEMBL27365433 0.78 KEAP1 (0.95) KEAP1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL11512295 0.78 KEAP1 (0.95) KEAP1LMNACYP1A2CYP2D6CYP2C9
Hydrogen Sulfide SCHEMBL27698561 0.78 KEAP1 (0.95) KEAP1LMNACYP1A2CYP2D6CYP2C9
Fluoride SCHEMBL28258745 0.78 KEAP1 (0.95) KEAP1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL21092440 0.76 KIF11 (0.69) KEAP1USP2LMNACYP1A2CYP3A4
SCHEMBL31041151 0.75 KIF11 (0.79) KEAP1LMNACYP2C9CLK4PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100263306-A1 ROOM WITH TWO COUNTER-RESISTANT INSECTICIDAL OBJECTS VESTERGAARD FRANDSEN SA (CH) 2010-10-21 US disclosed
EP-2219444-A2 ROOM WITH TWO COUNTER-RESISTANT INSECTICIDAL OBJECTS Vestergaard Frandsen SA (CH) 2010-08-25 EP disclosed
US-20100119720-A1 PROCESS FOR INSECTICIDAL IMPREGNATION OF A FABRIC OR NETTING OR OTHER KIND OF NON-LIVING MATERIAL VESTERGAARD FRANDSEN SA (CH) 2010-05-13 US disclosed
EP-2141987-A1 PROCESS FOR INSECTICIDAL IMPREGNATION OF A FABRIC OR NETTING OR OTHER KIND OF NON-LIVING MATERIAL Vestergaard Frandsen SA (CH) 2010-01-13 EP disclosed
WO-2009059603-A1 ROOM WITH TWO COUNTER-RESISTANT INSECTICIDAL OBJECTS VESTERGAARD FRANDSEN SA (CH) 2009-05-14 WO disclosed
WO-2009059607-A2 ROOM WITH TWO COUNTER-RESISTANT INSECTICIDAL OBJECTS VESTERGAARD FRANDSEN SA (CH) 2009-05-14 WO disclosed
WO-2008122287-A1 PROCESS FOR INSECTICIDAL IMPREGNATION OF A FABRIC OR NETTING OR OTHER KIND OF NON-LIVING MATERIAL VESTERGAARD FRANDSEN SA (CH) 2008-10-16 WO disclosed
CN-101247722-A Biphenyl-N- (4-pyridyl) methylsulfonamides BASF AG (DE) 2008-08-20 CN disclosed
US-20080161187-A1 Controlling phytopathogenic harmful fungi and harmful arthropodes; combating arthropodal pestsprotecting crops, seeds and non-living materials from infestation by arthropodal pests; insecticides, pesticides, fungicides; miticides; agriculture; veterinary medicine BASF AKTIENGESELLSCHAFT (DE) 2008-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161187-A1 Controlling phytopathogenic harmful fungi and harmful arthropodes; combating arthropodal pestsprotecting crops, seeds and non-living materials from infestation by arthropodal pests; insecticides, pesticides, fungicides; miticides; agriculture; veterinary medicine PTPN21, PTPN1, PTPN14 KEAP1 395/4885CYP17A1 1107/4885USP2 1093/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.