SCHEMBL28005209

SCHEMBL28005209

Cc1cc(Nc2ccccc2N)cc(C)c1Br

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
GAA P10253 4/20 0.58
TDP1 Q9NUW8 3/20 0.58
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 3/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
MAPK14 Q16539 11/20 0.52
MAPK13 O15264 9/20 0.52
MAPK12 P53778 9/20 0.52
MAPK11 Q15759 9/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
ALOX15 P16050 2/20 0.52
TP53 P04637 1/20 0.52
APP P05067 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9994865 0.83 MAPT (0.59) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL2931765 0.80 MAPT (0.74) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL5492276 0.80 MAPT (0.65) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL9183066 0.79 MAPT (0.69) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL2944533 0.79 MAPT (0.69) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL16532020 0.75 MAPT (0.49) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL4607773 0.74 MAPT (0.86) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL6563685 0.74 MAPK13 (0.54) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL2602405 0.73 MAPT (1.00) MAPTGAATDP1ALDH1A1KDM4E
SCHEMBL2764151 0.73 MAPT (0.70) MAPTGAATDP1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104418866-A DGAT1 inhibitor, and preparation method and application thereof NANJING MINGDE NEW DRUG RES AND DEV CO LTD 2015-03-18 CN disclosed