SCHEMBL28014367

SCHEMBL28014367

Cc1ccccc1-c1cc(C=O)cs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.39
ALDH1A1 P00352 5/20 0.38
TSHR P16473 1/20 0.38
ATP4A P20648 2/20 0.35
ATP4B P51164 2/20 0.35
CYP2A6 P11509 2/20 0.34
RAB9A P51151 5/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
KDM4E B2RXH2 2/20 0.33
MAOB P27338 2/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
PLA2G7 Q13093 1/20 0.32
NPC1 O15118 4/20 0.32
MAPK1 P28482 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27858647 0.79 CYP2A6 (0.34) ALDH1A1CYP2A6HTR2B
SCHEMBL27875009 0.78 ALDH1A1 (0.33) ALDH1A1CYP2A6HTR2B
SCHEMBL27858658 0.78 ALDH1A1 (0.33) ALDH1A1CYP2A6HTR2B
SCHEMBL723278 0.74 ALDH1A1 (0.44) ALDH1A1CYP2A6RAB9AKDM4EMAOB
SCHEMBL16012707 0.73 HPGD (0.39) HPGDALDH1A1TSHRATP4AATP4B
SCHEMBL28087582 0.71 HSD17B1 (0.42) HPGDALDH1A1TSHRCYP2A6RAB9A
SCHEMBL28014366 0.71 CYP2A6 (0.48) HPGDALDH1A1CYP2A6RAB9ASMN1; SMN2
SCHEMBL29291122 0.70 RAB9A (0.37) HPGDALDH1A1TSHRATP4AATP4B
SCHEMBL28057584 0.70 HPGD (0.44) HPGDALDH1A1TSHRRAB9ASMN1; SMN2
SCHEMBL16511765 0.70 ALDH1A1 (0.41) ALDH1A1CYP2A6SMN1; SMN2RXFP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103304555-B One group of benzene-oxazolyl derivative and preparation method thereof and the related application as IMPDH inhibitor INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-03-30 CN disclosed
CN-103442566-B The compound of Therapeutic cancer GTX, INC. (US) 2015-12-09 CN disclosed
CN-102883607-B Compounds for the treatment of cancer GTX INC 2015-07-22 CN disclosed
CN-104736530-A Compounds for the treatment of paramoxyvirus viral infections ALIOS BIOPHARMA INC 2015-06-24 CN disclosed
CN-104592205-A COMPOUNDS FOR TREATMENT OF CANCER GTX INC 2015-05-06 CN disclosed