SCHEMBL28019097

SCHEMBL28019097

O=C(O)c1cc(Cl)c(CCBr)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SCN9A Q15858 6/20 0.37
MRGPRX4 Q96LA9 3/20 0.37
KDM4E B2RXH2 2/20 0.35
ASPH Q12797 1/20 0.35
KDM8 Q8N371 1/20 0.35
ALDH1A1 P00352 3/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15018380 0.86 KEAP1 (0.41) KEAP1NFE2L2SCN9AMRGPRX4KDM4E
SCHEMBL15543742 0.81 KEAP1 (0.42) KEAP1NFE2L2SCN9AMRGPRX4KDM4E
SCHEMBL27979581 0.78 KDM1A (0.31)
SCHEMBL14331830 0.76 KEAP1 (0.50) KEAP1NFE2L2MRGPRX4KDM4EASPH
SCHEMBL363365 0.74 KEAP1 (0.48) KEAP1NFE2L2MRGPRX4KDM4EASPH
SCHEMBL29488312 0.74 KEAP1 (0.48) KEAP1NFE2L2MRGPRX4KDM4EASPH
SCHEMBL18420388 0.73 KDM4E (0.40) KEAP1NFE2L2MRGPRX4KDM4EASPH
SCHEMBL16618297 0.73 KEAP1 (0.44) KEAP1NFE2L2MRGPRX4KDM4EASPH
SCHEMBL28353593 0.72 HMGB1 (0.37) KDM4EALDH1A1TSHRHPGDHSD17B10
SCHEMBL16387317 0.71 DGAT1 (0.43) SCN9AALDH1A1CASP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104718188-A N-substituted benzamides and their use in the treatment of pain GENENTECH INC 2015-06-17 CN disclosed