SCHEMBL28020178

SCHEMBL28020178

O=C(c1c(Cl)cccc1C1CC1)c1c(Cl)cccc1C1CC1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 17/20 0.48
ALDH1A1 P00352 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
KMT2A Q03164 1/20 0.42
PPARG P37231 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15569345 0.87 ALDH1A1 (0.61) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL15569786 0.87 RORC (0.46) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL21181630 0.85 TAS1R3 (0.44) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL16888471 0.85 TAS1R3 (0.44) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL15565811 0.81 SLC6A3 (0.51) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL16981800 0.81 TAS1R3 (0.42) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL16884658 0.81 TAS1R3 (0.42) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL20275229 0.81 TAS1R3 (0.48) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL18810137 0.81 TAS1R3 (0.48) RORCALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL15570712 0.80 ALDH1A1 (0.57) RORCALDH1A1TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104853757-A 4-heteroaryl substituted benzoic acid compounds as ROR gamma T inhibitors and uses thereof MERCK SHARP & DOHME 2015-08-19 CN disclosed