SCHEMBL28020698

SCHEMBL28020698

COc1ccc(CC(=O)Nc2ccc(C(=O)NNC(=O)c3ccccc3)cc2)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
KMT2A Q03164 7/20 0.56
MEN1 O00255 6/20 0.56
BCHE P06276 4/20 0.55
ACHE P22303 4/20 0.55
POLB P06746 4/20 0.55
HPGD P15428 3/20 0.55
EPHX2 P34913 1/20 0.54
CYP3A4 P08684 1/20 0.54
KDM4E B2RXH2 5/20 0.53
TDP1 Q9NUW8 2/20 0.53
HTT P42858 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 2/20 0.53
NPSR1 Q6W5P4 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28020363 0.92 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2KMT2AMEN1BCHE
SCHEMBL28020357 0.90 BCHE (0.68) ALDH1A1SMN1; SMN2KMT2AMEN1BCHE
SCHEMBL28020735 0.87 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2KMT2AMEN1BCHE
SCHEMBL28020740 0.86 MEN1 (0.62) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL28020305 0.85 EPHX2 (0.58) ALDH1A1SMN1; SMN2KMT2ABCHEACHE
SCHEMBL29944814 0.78 ROCK2 (0.64) ALDH1A1SMN1; SMN2KMT2AMEN1HPGD
SCHEMBL28820179 0.77 MEN1 (0.52) ALDH1A1SMN1; SMN2KMT2AMEN1POLB
SCHEMBL21357031 0.77 NPC1 (0.74) ALDH1A1SMN1; SMN2KMT2AMEN1POLB
SCHEMBL3653095 0.77 EPHX2 (0.77) ALDH1A1SMN1; SMN2KMT2AMEN1BCHE
SCHEMBL28020302 0.77 EPHX2 (0.61) ALDH1A1SMN1; SMN2KMT2AMEN1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102775381-B Substituted hydrazide compound, and its preparation method, medicinal compositions and application SHANGHAI INST MATERIA MEDICA 2015-05-20 CN disclosed