SCHEMBL28020904

SCHEMBL28020904

COc1ccccc1Cc1sc(NCc2ccc(C#N)cc2)nc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.42
CYP1A2 P05177 4/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2C19 P33261 4/20 0.42
CLK4 Q9HAZ1 3/20 0.42
CYP2D6 P10635 3/20 0.42
MEN1 O00255 2/20 0.42
USP2 O75604 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 2/20 0.42
LMNA P02545 2/20 0.42
CYP2C9 P11712 1/20 0.42
NTRK1 P04629 1/20 0.42
NTRK3 Q16288 1/20 0.42
NTRK2 Q16620 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 3/20 0.41
PTGDR2 Q9Y5Y4 3/20 0.41
NPC1 O15118 2/20 0.41
ADORA2A P29274 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28020562 0.92 CYP1A2 (0.46) GAACYP1A2CYP3A4CYP2C19CLK4
SCHEMBL27907145 0.88 PTGDR2 (0.47) GAACYP1A2CYP3A4CYP2C19MEN1
SCHEMBL28020949 0.86 NPC1 (0.52) GAACLK4MEN1KMT2ATSHR
SCHEMBL27907174 0.85 LMNA (0.51) GAACYP1A2CYP3A4CYP2C19CLK4
SCHEMBL27925087 0.76 NPC1 (0.54) GAACLK4MEN1KMT2AALDH1A1
SCHEMBL4452157 0.74 KMT2A (0.42) GAAMEN1KMT2ALMNAPTGDR2
SCHEMBL27925165 0.71 CETP (0.50) GAACLK4MEN1KMT2AALDH1A1
SCHEMBL27907149 0.69 PTGDR2 (0.52) GAACYP3A4CYP2C19CYP2D6MEN1
SCHEMBL27907147 0.67 RAB9A (0.54) GAAMEN1KMT2ALMNAMAPK1
SCHEMBL1303890 0.67 ADORA1 (0.57) CYP2C19MEN1USP2KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103159695-B HIV can be suppressed to copy and to effective thiazole compound of resistance HIV virus strain and its production and use CAPITAL NORMAL UNIVERSITY (CN) 2015-08-12 CN claimed
CN-103159695-B HIV can be suppressed to copy and to effective thiazole compound of resistance HIV virus strain and its production and use CAPITAL NORMAL UNIVERSITY (CN) 2015-08-12 CN disclosed