SCHEMBL28020949

SCHEMBL28020949

COc1ccc(CNc2nc(-c3ccccc3)c(Cc3ccc(C#N)cc3)s2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.52
ALDH1A1 P00352 2/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PTGDR2 Q9Y5Y4 5/20 0.46
DYRK1A Q13627 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
RAB9A P51151 1/20 0.45
ADORA1 P30542 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
CETP P11597 1/20 0.44
VNN1 O95497 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27925087 0.90 NPC1 (0.54) NPC1ALDH1A1GAATP53MAPT
SCHEMBL28020904 0.86 GAA (0.42) NPC1ALDH1A1GAAKDM4ETP53
SCHEMBL28020562 0.86 CYP1A2 (0.46) ALDH1A1GAAKDM4EMAPTHPGD
SCHEMBL28804129 0.83 PLTP (0.52) NPC1ALDH1A1GAAMAPTHPGD
SCHEMBL27925165 0.83 CETP (0.50) NPC1ALDH1A1GAATP53MAPT
SCHEMBL27907145 0.81 PTGDR2 (0.47) NPC1ALDH1A1GAAKDM4EMAPT
SCHEMBL1303890 0.80 ADORA1 (0.57) NPC1MAPTPTGDR2RAB9AADORA1
SCHEMBL27907150 0.76 ADORA2A (0.50) NPC1ALDH1A1KDM4ETP53MAPT
SCHEMBL27907147 0.76 RAB9A (0.54) NPC1GAAKDM4ETP53MAPT
SCHEMBL1302328 0.74 PLTP (0.58) NPC1ALDH1A1KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103159695-B HIV can be suppressed to copy and to effective thiazole compound of resistance HIV virus strain and its production and use CAPITAL NORMAL UNIVERSITY (CN) 2015-08-12 CN claimed
CN-103159695-B HIV can be suppressed to copy and to effective thiazole compound of resistance HIV virus strain and its production and use CAPITAL NORMAL UNIVERSITY (CN) 2015-08-12 CN disclosed