SCHEMBL28021728

SCHEMBL28021728

CCc1ccnc(-c2cccc(Cl)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.53
CYP3A4 P08684 3/20 0.50
CYP2C19 P33261 1/20 0.50
CYP19A1 P11511 1/20 0.48
LMNA P02545 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
DHFR P00374 1/20 0.43
MAP4K4 O95819 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
KMO O15229 1/20 0.41
DYRK1A Q13627 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27285044 0.80 TRPV3 (0.55) CYP19A1LMNAKDM4EALDH1A1CYP1A2
SCHEMBL27135558 0.80 MAPT (0.42) CYP3A4CYP2C19LMNAKDM4EALDH1A1
SCHEMBL15661361 0.79 PDE4B (0.61) PDE4BCYP3A4CYP2C19LMNAKDM4E
SCHEMBL2299616 0.79 KMO (0.44) CYP1A2MAPTKMT2AKMODYRK1A
SCHEMBL17826980 0.79 CNR2 (0.47) PDE4BCYP3A4CYP2C19CYP19A1KDM4E
SCHEMBL2666351 0.79 CYP19A1 (0.51) CYP19A1TSHRMAP4K4MAPTRAB9A
SCHEMBL8344326 0.78 CYP19A1 (0.54) CYP19A1KDM4EALDH1A1TSHRDHFR
SCHEMBL28483259 0.76 KMO (0.59) CYP19A1KDM4ETSHRMAP4K4MAPT
SCHEMBL30271753 0.76 CYP19A1 (0.51) CYP19A1TSHRDHFRMAP4K4MAPT
SCHEMBL16629543 0.76 CTSS (0.50) PDE4BCYP3A4CYP2C19KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104768932-A Heteroaryl inhibitors of PDE4 TETRA DISCOVERY PARTNERS LLC 2015-07-08 CN disclosed