SCHEMBL28022016

SCHEMBL28022016

CC(C)(C)NC(=O)Oc1ccncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.37
P2RX7 Q99572 1/20 0.37
KDM4E B2RXH2 3/20 0.35
BRAF P15056 1/20 0.35
KDR P35968 1/20 0.35
MAPK14 Q16539 1/20 0.35
TNNI3K Q59H18 1/20 0.35
GAA P10253 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HSP90AA1 P07900 1/20 0.33
GPR119 Q8TDV5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10771231 0.79 TSHR (0.57) RAB9ASMN1; SMN2POLBTSHRKDM4E
SCHEMBL30606641 0.78 ELANE (0.43) P2RX7KDM4EALDH1A1HSP90AA1
SCHEMBL15911401 0.78 P2RX7 (0.51) P2RX7KDM4EBRAFKDRMAPK14
SCHEMBL6648327 0.76 P2RX7 (0.41) HPGDSMN1; SMN2P2RX7KDM4EBRAF
SCHEMBL3548849 0.76 RAB9A (0.46) RAB9AHPGDSMN1; SMN2POLBKDM4E
SCHEMBL12470613 0.75 HSP90AA1 (0.40) RAB9AHPGDSMN1; SMN2POLBTSHR
SCHEMBL5968188 0.75 ELANE (0.44) RAB9AP2RX7KDM4EBRAFKDR
SCHEMBL27851405 0.74 KDM4E (0.51) RAB9AHPGDSMN1; SMN2KDM4EGAA
SCHEMBL30575119 0.74 HSP90AA1 (0.39) RAB9AHPGDSMN1; SMN2POLBTSHR
SCHEMBL29080505 0.74 HSP90AA1 (0.39) RAB9AHPGDSMN1; SMN2POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110325516-A HETEROARYL COMPOUNDS AND THEIR USE 米尼奥尔克斯治疗有限公司 2019-10-11 CN disclosed
CN-108349963-A sodium channel blockers 株式会社大熊制药 2018-07-31 CN disclosed
CN-104854107-A Pyrrolopyrimidine compounds as kinase inhibitors PHARMACYCLICS INC 2015-08-19 CN disclosed