SCHEMBL28022353

SCHEMBL28022353

O=C(OCl)c1ccc(-c2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 1/20 0.47
SRD5A2 P31213 1/20 0.44
S1PR1 P21453 4/20 0.43
ADH5 P11766 1/20 0.43
AKR1C3 P42330 7/20 0.42
AKR1C2 P52895 7/20 0.42
AKR1C4 P17516 1/20 0.41
AKR1C1 Q04828 1/20 0.41
EGFR P00533 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
S1PR3 Q99500 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
PTGS2 P35354 1/20 0.39
NOTUM Q6P988 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3903631 0.85 EGFR (0.57) SRD5A2S1PR1AKR1C3AKR1C2AKR1C4
SCHEMBL27702486 0.83 AKR1C3 (0.50) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL402398 0.83 ADH5 (0.58) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL27724772 0.82 PDK2 (0.51) SRD5A2S1PR1AKR1C3AKR1C2
SCHEMBL403135 0.80 AKR1C3 (0.55) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL17133900 0.80 AKR1C3 (0.60) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL28022856 0.77 FFAR2 (0.45) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL28192342 0.77 PLK1 (0.57) FFAR2S1PR1AKR1C3AKR1C2S1PR3
SCHEMBL28098468 0.77 MAPT (0.54) FFAR2SRD5A2S1PR1ADH5AKR1C3
SCHEMBL18046185 0.75 MLYCD (0.47) FFAR2SRD5A2S1PR1ADH5AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed