SCHEMBL28022356

SCHEMBL28022356

O=C(O)c1ccc(-c2ccccc2)c(C(F)(F)F)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.45
CLCN2 P51788 2/20 0.43
ACLY P53396 3/20 0.43
PTPN1 P18031 2/20 0.42
AKR1C2 P52895 3/20 0.41
AKR1C1 Q04828 3/20 0.41
HNF4A P41235 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C8 P10632 1/20 0.40
FOLH1 Q04609 1/20 0.40
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
ALDH1A1 P00352 1/20 0.39
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2524408 0.85 PTPN1 (0.46) PDK2ACLYPTPN1AKR1C2AKR1C1
SCHEMBL5934445 0.82 HNF4A (0.54) PTPN1AKR1C2AKR1C1HNF4ACYP2C8
SCHEMBL27587157 0.82 PTPN1 (0.44) CLCN2ACLYPTPN1AKR1C2AKR1C1
SCHEMBL2805234 0.81 ACLY (0.46) ACLYPTPN1AKR1C2AKR1C1HNF4A
SCHEMBL3927795 0.79 CLCN2 (0.54) PDK2CLCN2ACLYPTPN1AKR1C2
SCHEMBL2174123 0.78 HNF4A (0.58) PTPN1AKR1C2AKR1C1HNF4AFOLH1
SCHEMBL21776979 0.78 NOTUM (0.56) CLCN2TSHRALDH1A1RXRARXRB
SCHEMBL31369080 0.77 ALDH1A1 (0.43) PDK2ACLYPTPN1AKR1C2AKR1C1
SCHEMBL27881031 0.77 SYK (0.41) ACLYPTPN1AKR1C2AKR1C1HNF4A
SCHEMBL2579402 0.76 TSHR (0.41) PDK2CLCN2ACLYTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102449-B Antiviral compound 豪夫迈·罗氏有限公司 2017-06-13 CN disclosed
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed
CN-102803238-B Oxadiazole Derivatives MERCK SERONO S.A. (CH) 2015-09-30 CN disclosed