SCHEMBL28022700

SCHEMBL28022700

CS(=O)(=O)c1cccc(-c2ccccc2F)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.51
SCD O00767 2/20 0.51
FADS1 O60427 1/20 0.51
KAT6A Q92794 1/20 0.50
PTPRC P08575 1/20 0.49
PTPN1 P18031 1/20 0.49
JAK2 O60674 2/20 0.47
FAAH O00519 1/20 0.46
PARP1 P09874 1/20 0.46
NR1H2 P55055 2/20 0.45
NR1H3 Q13133 2/20 0.45
JAK3 P52333 1/20 0.44
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30604310 0.85 HSD17B1 (0.47) PTGS2KAT6AJAK2FAAHPARP1
SCHEMBL4159024 0.83 BRD4 (0.55) SCDKAT6APTPRCPTPN1NR1H2
SCHEMBL308372 0.83 KAT6A (0.53) PTGS2KAT6APTPRCPTPN1BRD4
SCHEMBL14161390 0.83 CA1 (0.55) PTGS2SCDKAT6APTPRCPTPN1
SCHEMBL14120596 0.83 KAT6A (0.50) PTGS2SCDFADS1KAT6APTPRC
SCHEMBL17175626 0.81 FAAH (0.51) PTGS2KAT6AJAK2FAAHPARP1
SCHEMBL9206986 0.80 PTGS2 (0.73) PTGS2SCDFADS1
SCHEMBL25680126 0.80 JAK2 (0.45) PTGS2JAK2PARP1NR1H2NR1H3
SCHEMBL17165959 0.80 FAAH (0.42) PTGS2JAK2FAAHPARP1NR1H2
SCHEMBL28022794 0.79 NR1H2 (0.52) PTGS2SCDKAT6AJAK2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN claimed
CN-103443082-A Prodrugs of LXR modulating imidazole derivatives BRISTOL MYERS SQUIBB CO 2013-12-11 CN disclosed