SCHEMBL28022859

SCHEMBL28022859

O=C(O)C1CN2CCCC2[C@H]1C(=O)c1cccs1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ALDH1A1 P00352 2/20 0.44
SLC18A3 Q16572 5/20 0.44
KDM4E B2RXH2 1/20 0.41
THRB P10828 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 1/20 0.40
PABPC1 P11940 1/20 0.39
EIF4H Q15056 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27933965 0.75 ALDH1A1 (0.38) SMN1; SMN2ALDH1A1KDM4EL3MBTL1
SCHEMBL3858877 0.73 GAA (0.54) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL6201226 0.73 GAA (0.54) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL6201220 0.73 GAA (0.54) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL3866711 0.73 GAA (0.54) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL28022342 0.72 ALDH1A1 (0.38) NPC1RAB9AALDH1A1
SCHEMBL1578062 0.70 GAA (1.00) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL16615455 0.70 GAA (0.53) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL6290035 0.67 ALDH1A1 (0.60) GAAMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL6290034 0.67 ALDH1A1 (0.60) GAAMAPTSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703980-A Orexin receptor antagonists which are [ortho bi (hetero )aryl]-[2-(meta bi (hetero )aryl)-pyrrolidin-1-yl]-methanone derivatives ACTELION PHARMACEUTICALS LTD 2015-06-10 CN disclosed