SCHEMBL28022342

SCHEMBL28022342

O=C(O)C1CN2CCCC2[C@H]1C(=O)c1ccoc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
POLB P06746 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
CCR5 P51681 1/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
PTPN1 P18031 1/20 0.33
PTPN6 P29350 1/20 0.33
PTPN11 Q06124 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27933965 0.75 ALDH1A1 (0.38) ALDH1A1KMT2AMEN1POLB
SCHEMBL28022859 0.72 GAA (0.53) ALDH1A1NPC1RAB9A
SCHEMBL16463448 0.66 CA2 (0.56) ALDH1A1
SCHEMBL28022336 0.65 GPR119 (0.36) ALDH1A1KMT2AMEN1
SCHEMBL12449663 0.62 RECQL (0.63) ALDH1A1KMT2AMEN1POLBCHRNB2
SCHEMBL12986 0.62 RECQL (0.63) ALDH1A1KMT2AMEN1POLBCHRNB2
SCHEMBL19002209 0.62 RECQL (0.63) ALDH1A1KMT2AMEN1POLBCHRNB2
SCHEMBL13753568 0.61 GAA (0.62) ALDH1A1KMT2AMEN1POLBCHRNB2
SCHEMBL28159225 0.61 CHRNB2 (0.44) ALDH1A1KMT2AMEN1POLBCHRNB2
SCHEMBL11202198 0.61 CDC42 (0.59) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703980-A Orexin receptor antagonists which are [ortho bi (hetero )aryl]-[2-(meta bi (hetero )aryl)-pyrrolidin-1-yl]-methanone derivatives ACTELION PHARMACEUTICALS LTD 2015-06-10 CN disclosed