SCHEMBL28023906

SCHEMBL28023906

COc1ccc(CN2CNC(C(=O)C=O)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.46
MMP13 P45452 1/20 0.46
KDM4E B2RXH2 1/20 0.43
SIGMAR1 Q99720 2/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28367809 0.79 SIGMAR1 (0.47) MMP1MMP13KDM4ESIGMAR1SMN1; SMN2
SCHEMBL28808984 0.76 ACP1 (0.44) KDM4EHRH3SMN1; SMN2ALDH1A1
SCHEMBL2706345 0.71 MEN1 (0.46) SIGMAR1ALDH1A1
SCHEMBL23464746 0.71 MEN1 (0.46) SIGMAR1ALDH1A1
SCHEMBL203039 0.71 MEN1 (0.46) SIGMAR1ALDH1A1
SCHEMBL23540940 0.70 SIGMAR1 (0.49) MMP1MMP13KDM4ESIGMAR1POLB
SCHEMBL15532870 0.70 S1PR5 (0.69) KDM4ESIGMAR1
SCHEMBL2918073 0.69 SIGMAR1 (0.57) KDM4ESIGMAR1POLBSMN1; SMN2ALDH1A1
SCHEMBL5191850 0.68 LTA4H (0.49) KDM4ESIGMAR1POLBPKMHRH3
SCHEMBL23415558 0.68 S1PR5 (0.53) SIGMAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922347-A New imide derivative and its purposes as medicine 田边三菱制药株式会社 2018-04-17 CN disclosed
CN-102971291-B Novel amide derivative and use thereof as medicine MITSUBISHI TANABE PHARMA CORP 2015-07-22 CN disclosed