SCHEMBL28024329

SCHEMBL28024329

NC(=O)c1ccc2cncc(Cc3ccncc3)c2n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNC P24863 2/20 0.43
CDK8 P49336 2/20 0.43
CYP17A1 P05093 1/20 0.42
PIM1 P11309 2/20 0.40
NAMPT P43490 1/20 0.40
GRM2 Q14416 7/20 0.38
PNP P00491 1/20 0.38
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
PIM3 Q86V86 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
TSHR P16473 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28148153 0.83 PDE10A (0.44) CCNCCDK8GRM2
SCHEMBL28821086 0.82 CCNC (0.41) CCNCCDK8PIM1NAMPTGRM2
SCHEMBL28024317 0.78 CCNC (0.48) CCNCCDK8PIM1GRM2TSHR
SCHEMBL15741758 0.76 CCNC (0.46) CCNCCDK8PIM1HRH4
SCHEMBL28024785 0.76 CCNC (0.43) CCNCCDK8PIM1GRM2TSHR
SCHEMBL14266820 0.75 LMNA (0.41) CCNCCDK8
SCHEMBL28024769 0.74 CCNC (0.44) CCNCCDK8PIM1
SCHEMBL28821388 0.73 CCNC (0.44) CCNCCDK8PIM1
SCHEMBL1319809 0.71 CCNC (0.49) CCNCCDK8PIM1GRM2TSHR
SCHEMBL15742996 0.69 CCNC (0.62) CCNCCDK8PIM1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812387-A Substituted 1, 6-naphthyridines HOFFMANN LA ROCHE 2015-07-29 CN disclosed