SCHEMBL28148153

SCHEMBL28148153

COc1ccc(Cc2cncc3ccc(C(N)=O)nc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
CYP11B1 P15538 7/20 0.43
CYP11B2 P19099 7/20 0.43
GRM2 Q14416 5/20 0.43
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
MAP4K4 O95819 1/20 0.40
APP P05067 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024329 0.83 CCNC (0.43) GRM2CCNCCDK8
SCHEMBL28821086 0.82 CCNC (0.41) GRM2CYP2C9CCNCCDK8
SCHEMBL15742774 0.79 CCNC (0.65) CYP11B1CYP11B2GRM2CCNCCDK8
SCHEMBL28024769 0.77 CCNC (0.44) PDE10ACYP11B1CYP11B2CCNCCDK8
SCHEMBL4578523 0.76 PTGS1 (0.43) CYP11B1CYP11B2CCNCCDK8MAP4K4
SCHEMBL28148152 0.75 PDE10A (0.43) PDE10ACYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL28024317 0.73 CCNC (0.48) GRM2CCNCCDK8
SCHEMBL29670400 0.73 FTO (0.48) CYP11B1CYP11B2CYP19A1CYP2C9MAP4K4
SCHEMBL28024785 0.71 CCNC (0.43) GRM2CCNCCDK8
SCHEMBL28821388 0.71 CCNC (0.44) PDE10ACYP11B2CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106817900-A Novel naphthyridines and isoquinolin and its purposes as CDK8/19 inhibitor 默克专利有限公司 2017-06-09 CN disclosed