SCHEMBL28024317

SCHEMBL28024317

NC(=O)c1ccc2cncc(CCO)c2n1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNC P24863 10/20 0.48
CDK8 P49336 10/20 0.48
PIM1 P11309 2/20 0.43
DGAT1 O75907 3/20 0.36
ADORA3 P0DMS8 1/20 0.32
TSHR P16473 1/20 0.32
MC4R P32245 1/20 0.32
ADRA1A P35348 1/20 0.32
MC3R P41968 1/20 0.32
LCK P06239 1/20 0.31
TTK P33981 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
KMT2A Q03164 1/20 0.31
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024769 0.83 CCNC (0.44) CCNCCDK8PIM1
SCHEMBL28821388 0.82 CCNC (0.44) CCNCCDK8PIM1
SCHEMBL15741758 0.79 CCNC (0.46) CCNCCDK8PIM1
SCHEMBL28024785 0.79 CCNC (0.43) CCNCCDK8PIM1DGAT1ADORA3
SCHEMBL28024329 0.78 CCNC (0.43) CCNCCDK8PIM1TSHRGRM2
SCHEMBL1319809 0.74 CCNC (0.49) CCNCCDK8PIM1ADORA3TSHR
SCHEMBL28148153 0.73 PDE10A (0.44) CCNCCDK8GRM2
SCHEMBL4580346 0.73 CCNC (0.64) CCNCCDK8PIM1PIM2
SCHEMBL4729623 0.72 P2RX7 (0.44) CCNCCDK8ADORA3KMT2A
SCHEMBL4579667 0.72 CCNC (0.45) CCNCCDK8PIM1DGAT1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812387-A Substituted 1, 6-naphthyridines HOFFMANN LA ROCHE 2015-07-29 CN disclosed