SCHEMBL28026227

SCHEMBL28026227

C=C(C)c1cccc(F)n1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 5/20 0.38
MAPT P10636 2/20 0.37
CTSA P10619 2/20 0.35
KDM4E B2RXH2 2/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
ACMSD Q8TDX5 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CLK1 P49759 1/20 0.33
CLK2 P49760 1/20 0.33
HSD17B14 Q9BPX1 1/20 0.32
LMNA P02545 1/20 0.32
PAX8 Q06710 1/20 0.32
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13793158 0.84 KDM4E (0.46) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL2632248 0.78 ALDH1A1 (0.47) GRM4MAPTCTSAKDM4EALOX15
SCHEMBL24439792 0.78 GRM4 (0.39) GRM4MAPTCTSAKDM4EALOX15
SCHEMBL8281251 0.76 P2RX7 (0.50) GRM4CTSAKDM4EALOX15TSHR
SCHEMBL21615647 0.76 KDM4E (0.44) MAPTKDM4EALOX15TSHRACMSD
SCHEMBL13465025 0.74 KDM4E (0.33) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL21286483 0.74 KDM4E (0.38) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL9368741 0.74 ALDH1A1 (0.42) MAPTCTSAKDM4EALOX15TSHR
SCHEMBL8282746 0.74 NOS2 (0.46) GRM4KDM4EALOX15TSHRACMSD
SCHEMBL531659 0.74 GRM5 (0.44) MAPTCTSAKDM4EALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106117193-A New Hete rocyclic derivatives and the application in nervous system disease is treated thereof 诺华股份有限公司 2016-11-16 CN disclosed
CN-103403001-B Heterocyclic derivatives and their use in the treatment of neurological disorders 诺瓦提斯公司 2016-08-17 CN disclosed
CN-104955805-A Inhibitors of syk HOFFMANN LA ROCHE 2015-09-30 CN disclosed