SCHEMBL28026451

SCHEMBL28026451

COc1ccc(S(=O)(=O)c2ccc3c(c2)C(C)(C)CN3)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.51
GAA P10253 1/20 0.45
PTGIR P43119 1/20 0.41
RAPGEF4 Q8WZA2 1/20 0.41
HSD11B1 P28845 1/20 0.41
AKR1B1 P15121 1/20 0.41
CA2 P00918 2/20 0.40
HTR6 P50406 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ALDH1A1 P00352 1/20 0.39
RXRA P19793 1/20 0.39
HTT P42858 1/20 0.38
CYP26B1 Q9NR63 1/20 0.38
NFE2L2 Q16236 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8469485 0.81 PDE3B (0.45) GAAAKR1B1CA2PDE3BPDE3A
SCHEMBL15575858 0.77 RXRA (0.39) GAACA2ALDH1A1RXRACYP26B1
SCHEMBL15812262 0.73 HTR2C (0.46) GAAHTR6ALDH1A1HTTCYP26B1
SCHEMBL13074716 0.72 PKM (1.00) PKMGAARAPGEF4HSD11B1AKR1B1
SCHEMBL14486413 0.72 PKM (1.00) PKMGAARAPGEF4HSD11B1AKR1B1
SCHEMBL835692 0.72 PKM (1.00) PKMGAARAPGEF4HSD11B1AKR1B1
SCHEMBL9336566 0.70 MAPT (0.37) MEN1KMT2A
SCHEMBL17614163 0.68 PKM (0.52) PKMGAARAPGEF4HSD11B1CA2
SCHEMBL10497592 0.68 ALDH1A1 (0.63) PKMGAARAPGEF4CA2HTR6
SCHEMBL10828080 0.68 MEN1 (0.46) GAAALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103492376-B Bicyclic heterocycle compounds and their uses in therapy ASTEX THERAPEUTICS LTD 2015-07-22 CN disclosed