SCHEMBL28026689

SCHEMBL28026689

O=C(O)[C@H]1CC[C@H](C(=O)c2ncccc2SCc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
CYP2C9 P11712 1/20 0.45
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 4/20 0.41
PKM P14618 1/20 0.41
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 3/20 0.38
MAPT P10636 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
PTPRC P08575 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28026693 1.00 ALDH1A1 (0.45) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL2538269 0.87 L3MBTL1 (0.47) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL2538266 0.87 L3MBTL1 (0.47) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL28026658 0.80 KMT2A (0.52) ALDH1A1CYP2C9L3MBTL1KMT2AMEN1
SCHEMBL28026661 0.80 KMT2A (0.52) ALDH1A1CYP2C9L3MBTL1KMT2AMEN1
SCHEMBL3804451 0.80 ALDH1A1 (0.59) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL17022254 0.78 ALDH1A1 (0.50) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL28027191 0.77 CA12 (0.44) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL28027193 0.77 CA12 (0.44) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM
SCHEMBL13058357 0.75 HDAC6 (0.56) ALDH1A1CYP2C9HSD17B10L3MBTL1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102858778-B Heterobiaryl-cyclohexyl-tetrazine is [e] Azulene also HOFFMAN-LA ROCHE LTD. (CH) 2015-08-26 CN disclosed