SCHEMBL28027191

SCHEMBL28027191

O=C(O)[C@H]1CC[C@H](C(=O)c2ccncc2SCc2ccccc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ALDH1A1 P00352 3/20 0.39
CYP2C9 P11712 1/20 0.39
RAB9A P51151 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM6B O15054 3/20 0.38
KDM4C Q9H3R0 3/20 0.38
KDM4D Q6B0I6 2/20 0.38
KDM4E B2RXH2 1/20 0.38
KDM4A O75164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28027193 1.00 CA12 (0.44) CA12CA1CA2CA9CA14
SCHEMBL2542310 0.88 L3MBTL1 (0.41) CA12CA1CA2CA9CA14
SCHEMBL2542315 0.88 L3MBTL1 (0.41) CA12CA1CA2CA9CA14
SCHEMBL28026658 0.84 KMT2A (0.52) ALDH1A1CYP2C9RAB9AKMT2AGAA
SCHEMBL28026661 0.84 KMT2A (0.52) ALDH1A1CYP2C9RAB9AKMT2AGAA
SCHEMBL3776648 0.80 ALDH1A1 (0.54) CA12CA1CA2CA9CA14
SCHEMBL28026689 0.77 ALDH1A1 (0.45) CA12CA1CA2CA9CA14
SCHEMBL28026693 0.77 ALDH1A1 (0.45) CA12CA1CA2CA9CA14
SCHEMBL3785010 0.76 KMT2A (0.50) CA12CA1CA2CA9CA14
SCHEMBL3780022 0.74 L3MBTL1 (0.59) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102858778-B Heterobiaryl-cyclohexyl-tetrazine is [e] Azulene also HOFFMAN-LA ROCHE LTD. (CH) 2015-08-26 CN disclosed