SCHEMBL28028037

SCHEMBL28028037

CC1N=CC(O)(c2ccccc2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
POLB P06746 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
CCR2 P41597 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28028145 0.63 CHRNB2 (0.41) CRHBPCRHR2POLBGPR55ALDH1A1
SCHEMBL27954149 0.63 ALDH1A1 (0.35) POLBGPR55ALDH1A1SMN1; SMN2MEN1
SCHEMBL29531709 0.62 CRHBP (0.41) CRHBPCRHR2POLBALDH1A1MMP2
SCHEMBL27274817 0.61 POLB (0.39) POLBGPR55ALDH1A1SMN1; SMN2MEN1
SCHEMBL5924523 0.59 ALDH1A1 (0.47) POLBALDH1A1MMP2MMP9MEN1
SCHEMBL26342290 0.58 CCR2 (0.38) CRHBPCRHR2CCR2MEN1KMT2A
SCHEMBL2640739 0.58 MAPT (0.59) CHRNB2SLC6A2CHRNB4CHRNA3CHRNA4
SCHEMBL23375839 0.57 CCR2 (0.40) CRHBPCRHR2CHRNB2SLC6A2CHRNB4
SCHEMBL28806304 0.57 P2RX1 (0.35) SLC6A2SLC6A3
SCHEMBL21447355 0.57 CCR2 (0.40) CRHBPCRHR2CHRNB2SLC6A2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN claimed
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed