SCHEMBL28028675

SCHEMBL28028675

CS(=O)(=O)c1ccnc2[nH]ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 0.52
CHUK O15111 6/20 0.52
PRKCI P41743 3/20 0.50
AXL P30530 1/20 0.50
ROCK1 Q13464 2/20 0.45
PTK2 Q05397 2/20 0.45
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
PAK4 O96013 1/20 0.45
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
IGF1R P08069 1/20 0.45
FGFR1 P11362 1/20 0.45
PRKACA P17612 1/20 0.45
FLT1 P17948 1/20 0.45
LTK P29376 1/20 0.45
GRK5 P34947 1/20 0.45
KDR P35968 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12605441 0.83 TNNI3K (0.53) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL1075569 0.82 IKBKB (0.59) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL1036770 0.82 PRKCI (0.55) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL28111978 0.78 IKBKB (0.48) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL5137242 0.77 MET (0.64) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL7028646 0.75 IKBKB (0.49) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL4792437 0.74 IKBKB (0.74) IKBKBCHUKROCK1PTK2DAPK3
SCHEMBL3093132 0.72 PRKCI (0.55) IKBKBCHUKPRKCIAXLROCK1
SCHEMBL1701327 0.71 ADRA1A (0.34) IKBKBCHUKALK
SCHEMBL91443 0.71 PRKCI (0.59) IKBKBCHUKPRKCIAXLROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed