SCHEMBL28028823

SCHEMBL28028823

OCC(c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.44
CACNA1B Q00975 1/20 0.44
CACNB1 Q02641 1/20 0.44
CACNA1C Q13936 1/20 0.44
CYP19A1 P11511 3/20 0.44
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
ALDH1A1 P00352 2/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CNR2 P34972 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CRHBP P24387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980610 0.93 TRPA1 (0.43) CYP19A1LMNAHPGDCNR2TRPA1
SCHEMBL193835 0.85 HTR2A (0.52) LMNACYP2D6KDM4ETDP1HTR2A
Hydrochloric Acid SCHEMBL6251948 0.83 HTR2A (0.50) LMNACYP3A4CYP2D6KDM4ETDP1
Ammonia Solution, Strong SCHEMBL28352255 0.83 HTR2A (0.50) LMNACYP2D6KDM4ETDP1HTR2A
SCHEMBL6699187 0.83 CYP19A1 (0.49) CACNA2D1CACNA1BCACNB1CACNA1CCYP19A1
SCHEMBL21855514 0.79 CYP19A1 (0.51) CACNA1BCACNA1CCYP19A1LMNAHTT
SCHEMBL17814899 0.79 HTT (0.42) CYP19A1LMNAHTTNPSR1ALDH1A1
SCHEMBL11359363 0.79 CHRNB2 (0.61) LMNAALDH1A1HPGDCYP3A4CYP2D6
SCHEMBL7430169 0.77 CYP19A1 (0.44) CACNA2D1CACNA1BCACNB1CACNA1CCYP19A1
SCHEMBL7019079 0.77 CNR1 (0.49) CACNA2D1CACNA1BCACNB1CACNA1CCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104781256-B 3,4 pairs of substitution oxazolidinone derivatives and its purposes as the inhibitor of calcium-activated potassium channel 霍夫曼-拉罗奇有限公司 2017-09-29 CN disclosed
CN-104781256-A 3,4-disubstituted oxazolidinone derivatives and their use as inhibitors of the calcium activated potassium channel HOFFMANN LA ROCHE 2015-07-15 CN disclosed