SCHEMBL28028868

SCHEMBL28028868

COc1ccc(Cc2nc(N[C]=O)c3[nH]c(=O)n(Cc4ccccc4)c3n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.52
TLR7 Q9NYK1 10/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
HPGD P15428 2/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ADORA3 P0DMS8 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PNP P00491 1/20 0.44
MTOR P42345 1/20 0.43
ADORA2A P29274 1/20 0.43
IL6 P05231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28028872 0.78 TLR7 (0.49) NUDT1TLR7KDM4EALDH1A1HPGD
SCHEMBL19924572 0.71 TLR7 (0.47) NUDT1TLR7KDM4EALDH1A1HPGD
SCHEMBL23202278 0.70 TLR7 (0.57) NUDT1TLR7KDM4EALDH1A1HPGD
SCHEMBL28028891 0.70 ALDH1A1 (0.44) NUDT1TLR7KDM4EALDH1A1MAPT
SCHEMBL30011499 0.70 TLR7 (0.57) NUDT1TLR7KDM4EALDH1A1HPGD
SCHEMBL30012102 0.70 TRAP1 (0.69) TLR7KDM4EALDH1A1HPGDGAA
SCHEMBL23202316 0.70 TRAP1 (0.69) TLR7KDM4EALDH1A1HPGDGAA
SCHEMBL28029216 0.69 PIK3CD (0.49) NUDT1TLR7MTORADORA2A
SCHEMBL23392757 0.69 TLR7 (0.62) NUDT1TLR7KDM4EALDH1A1HPGD
SCHEMBL30012779 0.69 TLR7 (0.62) NUDT1TLR7KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107976546-A Inhibition of phosphorylation to TOR kinase inhibiting activities mark PRAS40, GSK3- β or P70S6K1 西格诺药品有限公司 2018-05-01 CN disclosed
CN-104870998-B inhibition of phosphorylation of PRAS40, GSK3- β or P70S6K1 as a marker of TOR kinase inhibitory activity 西格诺药品有限公司 2018-02-02 CN disclosed
CN-104870998-A Inhibition of phosphorylation of PRAS40, GSK 3-beta or P70S6K1 as a marker of TOR kinase inhibitory activity SIGNAL PHARM LLC 2015-08-26 CN disclosed