SCHEMBL28030659

SCHEMBL28030659

Clc1ccc(C2CN(Cc3ccccc3)CC2CNc2cnccn2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 5/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 1/20 0.42
RORC P51449 1/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
GRIN2B Q13224 1/20 0.39
SIGMAR1 Q99720 1/20 0.37
CNR2 P34972 1/20 0.37
KDM4E B2RXH2 1/20 0.36
DPP4 P27487 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
TACR2 P21452 1/20 0.35
TACR1 P25103 1/20 0.35
GBA1 P04062 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3025622 0.85 ALDH1A1 (0.43) CCR5ALDH1A1RORCSIGMAR1CNR2
SCHEMBL28030186 0.85 RORC (0.45) CCR5RORCGRIN2BSIGMAR1CNR2
SCHEMBL3025319 0.83 RORC (0.39) CCR5RORCSIGMAR1CNR2
SCHEMBL3029997 0.83 CCR5 (0.44) CCR5RORCSIGMAR1CNR2DPP4
SCHEMBL3029620 0.81 CCR5 (0.44) CCR5RORCSIGMAR1CNR2DPP4
SCHEMBL3019414 0.81 TACR1 (0.39) CCR5RORCCNR2TACR2TACR1
SCHEMBL3030612 0.79 CCR5 (0.46) CCR5ALDH1A1RORCSIGMAR1DPP4
SCHEMBL3031882 0.79 RORC (0.39) CCR5MEN1KMT2ARORCCYP3A4
SCHEMBL3032339 0.79 TACR1 (0.40) CCR5RORCGRIN2BSIGMAR1TACR2
SCHEMBL3032336 0.79 TACR1 (0.40) CCR5RORCGRIN2BSIGMAR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307853-B As the pyrrolidin derivatives of NK3 receptor antagonist F. HOFFMANN-LA ROCHE AG (CH) 2015-09-02 CN disclosed