SCHEMBL28031258

SCHEMBL28031258

CN(C)c1cccc(CC(N)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
KMT2A Q03164 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
ALDH1A1 P00352 4/20 0.46
TSHR P16473 1/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 2/20 0.44
CNR1 P21554 1/20 0.44
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GPR52 Q9Y2T5 1/20 0.43
AOC3 Q16853 1/20 0.41
CA2 P00918 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
KDM4E B2RXH2 2/20 0.41
NOS1 P29475 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2553049 0.84 KMT2A (0.54) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL3825118 0.84 HDAC1 (0.51) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL16009282 0.83 ALDH1A1 (0.51) KMT2AALDH1A1TSHRMAPK1MAPT
SCHEMBL6179341 0.83 ALDH1A1 (0.54) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL13378362 0.82 HTR3E (0.56) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL7259023 0.82 HDAC1 (0.50) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL10339219 0.80 CA2 (0.54) ALDH1A1MAPK1CA2KDM4ELMNA
SCHEMBL29844441 0.79 SLC7A5 (0.52) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL13865668 0.79 ALDH1A1 (0.43) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1
SCHEMBL27581167 0.78 HDAC1 (0.50) HDAC1HDAC6KMT2AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727307-A Compound and its application method 安吉奥斯医药品有限公司 2018-11-02 CN disclosed
CN-104936954-B Compounds and methods of use thereof 安吉奥斯医药品有限公司 2018-08-14 CN disclosed
CN-104936954-A compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2015-09-23 CN disclosed