SCHEMBL28032225

SCHEMBL28032225

COC(=O)c1c(-c2ccc([N+](=O)[O-])cc2)cn(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.46
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 3/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTPN11 Q06124 3/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
AURKA O14965 2/20 0.39
SLC6A3 Q01959 2/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28078513 0.88 MEN1 (0.49) KMT2AMEN1MAPTGAAHTT
SCHEMBL28031651 0.85 KMT2A (0.48) KMT2AMEN1MAPTGAAHTT
SCHEMBL28032238 0.84 SLC6A4 (0.47) KMT2AMEN1MAPTGAAHTT
SCHEMBL28031707 0.84 ALDH1A1 (0.46) KMT2AMEN1MAPTGAAHTT
SCHEMBL28032234 0.81 MEN1 (0.45) KMT2AMEN1MAPTGAAHTT
SCHEMBL28031631 0.80 PTPN11 (0.47) KMT2AMEN1MAPTPTPN11ALDH1A1
SCHEMBL28031624 0.80 GAA (0.46) KMT2AMEN1MAPTGAAHTT
SCHEMBL28031775 0.78 TP53 (0.45) KMT2AMEN1MAPTGAASMN1; SMN2
SCHEMBL28031622 0.78 KMT2A (0.43) KMT2AMEN1MAPTGAAHTT
SCHEMBL28032232 0.78 HTT (0.42) ARKMT2AMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017126-B Perfluoroalkyl azole derivatives and its synthetic method 上海麦克林生化科技有限公司 2018-01-19 CN disclosed
CN-105646322-A Perfluoroalkyl pyrrole derivative and synthesis method thereof 上海大学 2016-06-08 CN disclosed
CN-105017126-A Perfluoroalkyl pyrrole derivative and synthesis method thereof UNIV SHANGHAI 2015-11-04 CN disclosed