SCHEMBL28032950

SCHEMBL28032950

NC(c1cc(F)c(F)cc1F)[C@@H](CC(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TDP1 Q9NUW8 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
ALDH1A1 P00352 5/20 0.38
LTA4H P09960 3/20 0.38
LMNA P02545 2/20 0.38
SLC15A1 P46059 2/20 0.38
LAP3 P28838 1/20 0.38
IDO1 P14902 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28284788 1.00 DPP4 (0.41) DPP4KMT2ASMN1; SMN2TDP1SLC6A2
SCHEMBL28055241 0.77 DPP4 (0.37) DPP4
SCHEMBL27501468 0.77 ALDH1A1 (0.51) KMT2ASMN1; SMN2TDP1SLC6A2SLC6A3
SCHEMBL28937621 0.77 FFAR1 (0.33) DPP4TDP1
SCHEMBL28321679 0.76 SLC1A3 (0.54) KMT2ASMN1; SMN2TDP1SLC6A2SLC6A3
SCHEMBL29619670 0.73 DPP4 (0.49) DPP4ALDH1A1LTA4HLAP3
SCHEMBL11232982 0.72 DPP4 (0.51) DPP4KMT2AALDH1A1LTA4HSLC15A1
SCHEMBL28032955 0.72 DPP4 (0.51) DPP4KMT2AALDH1A1LTA4HSLC15A1
SCHEMBL27943329 0.72 DPP4 (0.51) DPP4KMT2AALDH1A1LTA4HSLC15A1
SCHEMBL10277201 0.72 CASP1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294479-A Preparation method of 3R-amino substituted butyrylamide derivative XINFA PHARMACEUTICAL CO LTD 2016-02-03 CN disclosed
CN-105061434-A Low-cost preparation method of sitagliptin phosphate XINFA PHARMACEUTICAL CO LTD 2015-11-18 CN disclosed