SCHEMBL28033083

SCHEMBL28033083

O=C(O)Cc1nccnc1Oc1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
TRPA1 O75762 2/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK14 Q16539 1/20 0.41
S1PR2 O95136 2/20 0.40
LTA4H P09960 1/20 0.40
FFAR1 O14842 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPBWR1 P48145 1/20 0.39
MCHR1 Q99705 1/20 0.39
HAO1 Q9UJM8 1/20 0.39
P2RY1 P47900 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28031196 0.83 FFAR1 (0.44) KMT2AFFAR1ALDH1A1SMN1; SMN2HAO1
SCHEMBL28822439 0.79 CXCL8 (0.56) ALDH1A1SMN1; SMN2
SCHEMBL28035897 0.76 KMT2A (0.47) KMT2ATRPA1CYP3A4MAPK14SMN1; SMN2
SCHEMBL28033082 0.72 CYP1A2 (0.43) KMT2ATRPA1CYP3A4MAPK14LTA4H
SCHEMBL3500048 0.72 SRD5A2 (0.62) KMT2AS1PR2LTA4HFFAR1
SCHEMBL28018126 0.72 GABRR1 (0.42) ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL2779361 0.71 KMT2A (0.65) KMT2AALDH1A1
SCHEMBL7371142 0.70 KMT2A (0.59) KMT2AALDH1A1
SCHEMBL9486549 0.69 CAMK2A (0.48) FFAR1ALDH1A1CYP1A2
SCHEMBL27566728 0.68 SCN9A (0.54) KMT2ALTA4HFFAR1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104961690-A Preparation method of 3-(4-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN disclosed
CN-104961691-A Preparation method of 3-(2-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN disclosed