SCHEMBL28033082

SCHEMBL28033082

CC(=O)Oc1nccnc1Oc1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
TRPA1 O75762 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAOB P27338 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAPK14 Q16539 1/20 0.40
LTA4H P09960 2/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8143090 0.83 TDP1 (0.53) CYP3A4CYP2C9KMT2APDE4AKDM4E
SCHEMBL7001893 0.83 KMT2A (0.49) CYP1A2CYP3A4TRPA1CYP2C9CYP2C19
SCHEMBL28031195 0.82 P2RY1 (0.42) CYP1A2CYP3A4CYP2C19KMT2AMAOB
SCHEMBL28822437 0.79 MAPT (0.46) TRPA1KMT2ASMN1; SMN2KDM4EMAPT
SCHEMBL28035897 0.75 KMT2A (0.47) CYP1A2CYP3A4TRPA1CYP2C9CYP2C19
SCHEMBL7674701 0.75 KMT2A (0.64) CYP1A2CYP2C9CYP2C19KMT2APDE4A
SCHEMBL660921 0.74 LMNA (0.64) CYP3A4KMT2ASMN1; SMN2MAOBKDM4E
Ammonia Solution, Strong SCHEMBL4479019 0.73 LMNA (0.61) CYP3A4KMT2ASMN1; SMN2MAOBKDM4E
Hydrochloric Acid SCHEMBL28555259 0.73 LMNA (0.61) CYP3A4KMT2ASMN1; SMN2MAOBKDM4E
SCHEMBL11578278 0.73 LMNA (0.61) CYP3A4KMT2ASMN1; SMN2MAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104961690-A Preparation method of 3-(4-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN disclosed
CN-104961691-A Preparation method of 3-(2-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN disclosed