SCHEMBL28033110

SCHEMBL28033110

NC(=O)c1ccc(-c2ccc(O)cc2)cc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPM1B O75688 1/20 0.54
IKBKB O14920 1/20 0.53
ESR2 Q92731 4/20 0.48
HSD17B1 P14061 2/20 0.46
CHUK O15111 1/20 0.46
ESR1 P03372 5/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
FYN P06241 1/20 0.43
KDM4E B2RXH2 2/20 0.42
GFER P55789 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ALOX5 P09917 1/20 0.42
PRF1 P14222 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HSP90AA1 P07900 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3781502 0.86 IKBKB (0.55) PPM1BIKBKBESR2CHUKKMT2A
SCHEMBL3793566 0.85 IKBKB (0.73) PPM1BIKBKBCHUKKMT2AMEN1
SCHEMBL6851164 0.85 PPM1B (0.74) PPM1BESR2HSD17B1KMT2AMEN1
SCHEMBL164897 0.84 CA12 (0.46) PPM1BIKBKBKMT2AMEN1KDM4E
SCHEMBL7281430 0.79 MKNK2 (0.58) IKBKBESR2HSD17B1CHUKESR1
SCHEMBL3784526 0.78 IKBKB (0.54) PPM1BIKBKBMEN1PRF1MKNK1
SCHEMBL23499274 0.75 PPM1B (0.79) PPM1BIKBKBESR2KMT2AMEN1
SCHEMBL29908977 0.75 PPM1B (0.79) PPM1BIKBKBESR2KMT2AMEN1
SCHEMBL7064896 0.75 ESR1 (0.43) ESR2HSD17B1CHUKESR1KDM4E
SCHEMBL20788509 0.75 IKBKB (0.55) IKBKBESR2CHUKESR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104955826-A SPIRO-QUINAZOLINONE DERIVATIVES USEFUL FOR THE TREATMENT OF NEUROLOGICAL DISEASES AND CONDITIONS MERCK PATENT GMBH 2015-09-30 CN disclosed