SCHEMBL28033876

SCHEMBL28033876

COc1cccc2c1ccc(=O)n2CCO

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 4/20 0.40
MTNR1A P48039 3/20 0.40
KCNA3 P22001 1/20 0.40
HTR2C P28335 1/20 0.40
CCR2 P41597 1/20 0.39
DAO P14920 1/20 0.39
CYP19A1 P11511 1/20 0.39
NQO2 P16083 1/20 0.39
GAA P10253 1/20 0.39
HTR6 P50406 1/20 0.39
CYP2A6 P11509 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8844829 0.83 KCNA3 (0.46) MTNR1BMTNR1AKCNA3HTR2CCCR2
SCHEMBL2797897 0.82 ALDH1A1 (0.51) MAPT
SCHEMBL2800336 0.79 TNFRSF1A (0.43) MTNR1BMTNR1AKCNA3HTR2CCCR2
SCHEMBL2798034 0.78 CCR2 (0.39) MTNR1BMTNR1AHTR2CCCR2HTR6
SCHEMBL17576252 0.78 KDM4E (0.49) KCNA3HTR2CCYP19A1NQO2GAA
SCHEMBL2799840 0.77 HTR6 (0.47) CCR2CYP19A1NQO2GAAHTR6
SCHEMBL9499742 0.76 DAO (0.51) HTR2CDAOCYP19A1NQO2GAA
SCHEMBL11999979 0.74 KDM4E (0.44) CYP19A1NQO2GAAMAPT
SCHEMBL7958454 0.74 HTR2C (0.60) HTR2CHTR6
SCHEMBL2795704 0.71 CYP19A1 (0.37) CCR2CYP19A1NQO2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105367583-A THIENO[2, 3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH 2016-03-02 CN disclosed
CN-102459280-B Thieno [2,3-b ] pyridine derivatives as inhibitors of viral replication KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2015-10-14 CN disclosed