SCHEMBL280357

SCHEMBL280357

Cc1cc(C)c(S(=O)(=O)CNc2cccnc2)s1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 2/20 0.41
ALPL P05186 8/20 0.41
LMNA P02545 2/20 0.40
NOTUM Q6P988 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.38
NAMPT P43490 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279726 0.80 NAMPT (0.46) ALDH1A1TP53TDP1RAB9AKMT2A
SCHEMBL10503692 0.69 SMN1; SMN2 (0.47) ALDH1A1TP53TDP1RAB9AKMT2A
SCHEMBL10503680 0.69 CA12 (0.62) ALDH1A1TP53TDP1RAB9AKMT2A
SCHEMBL12195638 0.68 NAMPT (0.65) TP53RAB9ALMNANAMPT
SCHEMBL2441007 0.67 RAB9A (0.53) RAB9ALMNANOTUMPOLBNAMPT
SCHEMBL1355489 0.64
Hydrochloric Acid SCHEMBL10704335 0.63 RAB9A (0.56) ALDH1A1RAB9ALMNAPOLBMAPK1
Hydrochloric Acid SCHEMBL28089121 0.63 RAB9A (0.56) ALDH1A1RAB9ALMNAPOLBMAPK1
SCHEMBL6739276 0.62 LMNA (0.56) ALDH1A1TP53TDP1KMT2AALPL
SCHEMBL790282 0.62 NAMPT (0.65) ALDH1A1TP53TDP1KMT2AALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134013-B2 Amide compound and thrombopoietin receptor activator NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-03-13 US disclosed
US-8134013-B2 Amide compound and thrombopoietin receptor activator NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-03-13 US disclosed
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-05-21 US disclosed
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-05-21 US disclosed
EP-1845090-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR Nissan Chemical Industries, Ltd. (JP) 2007-10-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR TEK, PTAFR, MPL ALDH1A1 2047/4885TP53 1466/4885TDP1 2969/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.