SCHEMBL28036066

SCHEMBL28036066

O=c1[nH]cnc2ccc(-c3ccccc3CO)cc12

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 7/20 0.64
TGFBR1 P36897 1/20 0.57
PARP1 P09874 6/20 0.53
PDPK1 O15530 1/20 0.53
CA12 O43570 1/20 0.53
ALOX15 P16050 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CA9 Q16790 1/20 0.53
TNKS2 Q9H2K2 1/20 0.53
IP6K1 Q92551 5/20 0.51
IP6K3 Q96PC2 4/20 0.51
IP6K2 Q9UHH9 3/20 0.51
CHEK1 O14757 1/20 0.48
PIM1 P11309 1/20 0.48
AKT1 P31749 1/20 0.48
FLT3 P36888 1/20 0.48
PIM3 Q86V86 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3740005 0.81 ACVR1 (0.74) ACVR1TGFBR1PARP1PDPK1CA12
SCHEMBL7980737 0.78 ACVR1 (0.67) ACVR1TGFBR1PARP1PDPK1CA12
SCHEMBL8622180 0.78 ACVR1 (0.73) ACVR1PARP1PDPK1CA12ALOX15
SCHEMBL18712269 0.75 ACVR1 (0.69) ACVR1TGFBR1PARP1PDPK1CA12
SCHEMBL9272871 0.75 ACVR1 (0.56) ACVR1TGFBR1PARP1PDPK1CA12
SCHEMBL7976876 0.75 TGFBR1 (0.58) ACVR1TGFBR1PARP1IP6K1IP6K3
SCHEMBL22980875 0.74 IP6K1 (0.66) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL28224560 0.74 IP6K1 (0.62) ACVR1PARP1IP6K1IP6K3IP6K2
SCHEMBL12304875 0.74 PARP1 (0.53) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL3731351 0.73 ACVR1 (0.60) ACVR1TGFBR1PARP1PDPK1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903300-A Comt inhibitors HOFFMANN LA ROCHE 2015-09-09 CN claimed
CN-104903300-A Comt inhibitors HOFFMANN LA ROCHE 2015-09-09 CN disclosed