SCHEMBL28036196

SCHEMBL28036196

COc1ccc(-c2ccccc2F)c(C(=O)O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.60
KDM4E B2RXH2 4/20 0.51
PRKAB2 O43741 1/20 0.49
PRKAG1 P54619 1/20 0.49
PRKAA2 P54646 1/20 0.49
PRKAA1 Q13131 1/20 0.49
PRKAG3 Q9UGI9 1/20 0.49
PRKAG2 Q9UGJ0 1/20 0.49
PRKAB1 Q9Y478 1/20 0.49
PTPN11 Q06124 1/20 0.49
POLB P06746 3/20 0.49
AKR1C3 P42330 2/20 0.48
AKR1C2 P52895 2/20 0.48
EIF4E P06730 1/20 0.47
GPR35 Q9HC97 1/20 0.47
GRM2 Q14416 1/20 0.47
ACMSD Q8TDX5 1/20 0.47
RAB9A P51151 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4600243 0.88 PRKAB2 (0.55) SMN1; SMN2KDM4EPRKAB2PRKAG1PRKAA2
SCHEMBL29853676 0.85 SMN1; SMN2 (0.79) SMN1; SMN2KDM4EPOLBAKR1C3AKR1C2
SCHEMBL7267474 0.85 SMN1; SMN2 (0.79) SMN1; SMN2KDM4EPOLBAKR1C3AKR1C2
SCHEMBL6536172 0.83 SMN1; SMN2 (0.62) SMN1; SMN2KDM4EPTPN11POLBAKR1C3
SCHEMBL5342329 0.81 SMN1; SMN2 (0.84) SMN1; SMN2KDM4EPOLBAKR1C3AKR1C2
SCHEMBL22537008 0.80 NPC1 (0.55) SMN1; SMN2KDM4EGRM2RAB9ANPC1
SCHEMBL14397805 0.80 SMN1; SMN2 (0.58) SMN1; SMN2KDM4EPTPN11POLBAKR1C3
SCHEMBL6574617 0.80 LMNA (0.53) SMN1; SMN2KDM4ERAB9ANPC1ALDH1A1
SCHEMBL2552037 0.79 SMN1; SMN2 (0.57) SMN1; SMN2KDM4EPTPN11POLBAKR1C3
SCHEMBL2313208 0.79 KDM4E (0.54) SMN1; SMN2KDM4EPRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903300-B COMT inhibitor 霍夫曼-拉罗奇有限公司 2018-04-17 CN disclosed
CN-104903300-A Comt inhibitors HOFFMANN LA ROCHE 2015-09-09 CN disclosed